Professional athletes and bodybuilders have been utilizing steroids for muscle growth and improved athletic performance for a long time.
However, they gradually discovered the detrimental implications that the steroids had. They were causing organ failures, sudden death, and a myriad of other severe medical complications. This made steroids too risky to justify the benefits.
People wanted a safer alternative.
Radius Health, Inc., a pharmaceutical company, developed “Testolone RAD 140,” also known as “Testolone,” to address this issue.
RAD 140 is a form of SARM (Selective Androgenic Receptor Modulator) under investigation that has all of the favorable effects of an anabolic steroid but none of the negative ones.
It was created to prevent muscle atrophy and is currently in the research stage. Still, many experts feel it has the potential to be utilized as a treatment for a variety of health issues in the future, including breast cancer.
People may wonder why they should utilize SARMs instead of steroids. The fundamental explanation for this is that SARMs are exceedingly selective when targeting androgenic receptors.
They target the androgen receptors in the bone and muscle tissues alone, whereas steroids interact with different organs.
Androgens are found in varying amounts in both male and female bodies. It is a natural hormone that aids in developing masculine traits and the regulation of secondary sex organ growth.
Testosterone is the primary androgen found in large amounts in males and affects masculine characteristics and reproductive activity.
SARMs mimic androgen effects by directly binding to androgen receptors. SARMs are extremely sensitive in their application and provide the most outstanding results.
On the other hand, steroids can be toxic at times, causing health issues such as liver damage, male breast enlargement, and abnormal hair growth in various places of the body in both men and women.
Even SARMs’ side effects pale in comparison to the side effects of steroids. This explains why bodybuilders and athletes love the RAD 140 supplement.
The structure of RAD 150, also known as TLB 150 or RAD 140 ester, is similar to that of rad-140. Its main chemical, RAD 140, was developed by Radius Health, INC. Due to its esterification during chemical production, RAD 150 is classed as an anabolic ester.
Esterification is the process of attaching ester groups to a carbon-based molecule, which is a frequent functional alteration. Chemical synthesis chemists have utilized it since the discovery of the first androgens.
This method is used to aid in the stabilization, enhancement, and modification of androgen bioavailability. This leads to a 10-fold increase in half-life, which is ten times longer than typical. This has resulted in a reduction in dosage frequency and an inconsistent hormone response in RAD 150.
Anabolic steroids had a lot of adverse effects before they were esterified. An increase in red blood cells, urine retention, and adverse effects on lipid profiles and the prostate gland are examples of this.
Esterification of testosterone, such as RAD 150, is now being studied in the hopes of stabilizing serum testosterone levels and reducing severe adverse effects.
SARM (Selective Androgen Receptor Modulator) research and development are now using this technology. Synthetic chemists are currently working on serum SARM levels to make them more stable and long-lasting.
The safety profiles of anabolic esters have improved in recent years. A variety of anabolic esters are currently being used to treat a variety of ailments. Nandrolone decanoate, for example, is administered to people with kidney failure, osteoporosis, and children with growth failure. The most widely administered anabolic-androgenic steroid is nandrolone decanoate. This is owing to the fact that it has a very long half-life in the body. Hair loss, acne shrinkage, gynecomastia, and testicular atrophy are the only drawbacks of nandrolone decanoate.
Testosterone undecanoate, another esterified version of testosterone, has also been used to treat metabolic disorders. This includes males who have low or no testosterone as a result of other medical issues. It aids in the development and maintenance of masculine sex features like body hair and a deep voice. It also has the added benefit of bringing plasma testosterone levels back to normal. Unfortunately, it has the same adverse side effects as nandrolone decanoate.
RAD 150 is the most efficient anabolic ester when compared to other anabolic esters. It provides positive outcomes while avoiding all of the undesirable side effects. It provides the body with longer-lasting pharmacokinetics, which means it is more effective in moving across the body.
This has attracted the research community’s curiosity greatly. When testosterone levels are elevated, they become more stable, lowering the chance of behavioral changes. It also rapidly attaches to the androgen receptor, causing it to become activated.
It has a great absorption rate and tissue-selective pharmacological patterns. As a result, rad 150 can provide a wide range of benefits. It also works as a buffer due to its long half-life.
RAD-150 continues to pique interest in biological research. This is partly owing to its potential to have an impact not just on the fitness community but also on the treatment of cancer and other metabolic disorders.
Due to its high absorption rate, stability, and 48-hour half-life, Rad 150 provides a wide range of benefits. At the same time, it has few to no adverse effects, especially when used as directed. This will be covered in more detail later in the article.
The following are some of the many advantages that rad 150 has to offer in terms of improving your performance and physique.
- It improves the body’s bone density and general muscle strength.
- RAD 150 can also be used to trim fat. It aids weight loss by melting down the fats deposited in the body.
- It raises the testosterone level in the body. Humans have a sense of enthusiasm and excitement when their testosterone levels are higher and their sexual desires are heightened. This is excellent for those suffering from sexual desire problems. High t-levels are also crucial for muscle building.
- It boosts the body’s muscle power and energy levels. Users are inspired and compelled to lift huge weights and do difficult tasks with ease. It delays fatigue and enhances recovery after each workout session.
- Memory and other functioning of the brain are destroyed by a protein called amyloid-beta. Testolone protects brain cells by preventing this protein from entering and improves the brain’s memory and learning capacity by promoting brain cell growth. It will also protect the brain from memory loss, which is expected as people age.
- RAD 150 inhibits the development of a protein known as ESR1, one of the components involved in breast cancer activation.
- It has no adverse effects on vital organs such as the liver and kidneys.
There are rarely any negative effects when the correct dosage is used. However, exceeding the recommended amount can result in a considerable increase in estradiol levels in the body.
Its great aromatizing action is the reason for this.
It can cause gynecomastia, a loss of muscular definition, and water retention under the skin. Headaches, sleeplessness, and extended erections are all possible side effects.
These side effects can be observed again if you take more than the advised dosage.
Although it does not cause liver damage, research is currently ongoing. Rad 150 is now being studied to see if it affects liver enzymes. It hasn’t been linked to any detrimental effects on the kidneys or prostate, thankfully.
Take two to three capsules twice a day. The dosages should be split throughout the day.
Rad 150 has a half-life of about 48 hours, which means it will be active in the body for about two days.
Post-cycle therapy (PCT) is always suggested towards the end of the cycle. Clomid, Arjuna, Coletix, and LiveR are just a few examples of good products you can use here. They will aid in restoring normal testosterone function, preserving lean muscle mass, and avoiding negative repercussions.
The TLB-150 is an updated version of the RAD-140. It does not, however, come from the creators of the latter. The term RAD-150 is derived from the structural resemblance of the two. TLB-150 is an “anabolic ester,” which means it boosts testosterone for longer than RAD-140. Indeed, its half-life is roughly 48 hours, whereas RAD-140’s is 16-18 hours. Because RAD-150 is accessible for extended periods, its effects are substantially more effective overall.
Not only that, but because it is esterified, RAD-150 is far more stable when it comes to raising Testosterone levels than other SARMs like MK-2866, RAD-140, and LGD-4033. RAD-150 minimizes the danger of behavioral changes such as increased aggression and removes male baldness and gynecomastia hazards by operating in this manner.
TLB-150 (RAD-150), although being relatively new to the market, is already vying for the top rank as the most effective SARM.